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Found 72 with Last Name = 'ruchala' and Initial = 'p'
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061360(CHEMBL3393878)
Affinity DataEC50:  1.10nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061361(CHEMBL3393877)
Affinity DataEC50:  8.40nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061362(CHEMBL3393876)
Affinity DataEC50:  10nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061363(CHEMBL3393875)
Affinity DataEC50:  34nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061364(CHEMBL3393874)
Affinity DataEC50:  218nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061365(CHEMBL3393873)
Affinity DataEC50:  13nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061366(CHEMBL3393872)
Affinity DataEC50:  10nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061367(CHEMBL3393871)
Affinity DataEC50:  6.30nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50061368(CHEMBL3393870)
Affinity DataEC50:  4.20nMAssay Description:Induction of human ferroportin degradation expressed in HEK293 cells after 24 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120919(CHEMBL3621383)
Affinity DataEC50:  300nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120920(CHEMBL3621379)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120949(CHEMBL3621380)
Affinity DataEC50:  458nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120950(CHEMBL3621378)
Affinity DataEC50:  52nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120951(CHEMBL3621377)
Affinity DataEC50:  369nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120952(CHEMBL3621376)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120953(CHEMBL3621375)
Affinity DataEC50:  92nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120954(CHEMBL3621374)
Affinity DataEC50:  165nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120955(CHEMBL3621373)
Affinity DataEC50:  269nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120956(CHEMBL3621372)
Affinity DataEC50:  335nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120957(CHEMBL3621371)
Affinity DataEC50:  113nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120958(CHEMBL3621370)
Affinity DataEC50:  104nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120959(CHEMBL3623073)
Affinity DataEC50:  44nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120960(CHEMBL3623072)
Affinity DataEC50:  75nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120961(CHEMBL3623071)
Affinity DataEC50:  54nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120962(CHEMBL3623070)
Affinity DataEC50:  532nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120963(CHEMBL3623069)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120964(CHEMBL3623068)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120965(CHEMBL3623067)
Affinity DataEC50:  517nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120966(CHEMBL3623066)
Affinity DataEC50:  477nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120967(CHEMBL3623065)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120968(CHEMBL3623064)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120969(CHEMBL3623063)
Affinity DataEC50:  599nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120970(CHEMBL3623062)
Affinity DataEC50:  272nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120971(CHEMBL3623061)
Affinity DataEC50:  586nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120972(CHEMBL3623060)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120988(CHEMBL3623059)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120989(CHEMBL3623058)
Affinity DataEC50: >600nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 40 member 1(Homo sapiens (Human))
University Of California Los Angeles

Curated by ChEMBL
LigandPNGBDBM50120990(CHEMBL3623057)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at GFP-fused human FPN transfected in HEK293 cells assessed as protein degradation after 24 hrs by flow cytometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500775(CHEMBL3758845)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at recombinant human NMU2 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500776(CHEMBL3759206)
Affinity DataEC50:  12nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500777(CHEMBL3759408)
Affinity DataEC50:  162nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500778(CHEMBL4299263)
Affinity DataEC50:  1.35E+3nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500779(CHEMBL3758577)
Affinity DataEC50:  0.214nMAssay Description:Agonist activity at recombinant human NMU2 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500780(CHEMBL3759820)
Affinity DataEC50:  43nMAssay Description:Agonist activity at recombinant human NMU2 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500781(CHEMBL3759626)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at recombinant human NMU2 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500782(CHEMBL3758687)
Affinity DataEC50:  56nMAssay Description:Agonist activity at recombinant human NMU2 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500783(CHEMBL3759452)
Affinity DataEC50:  0.575nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500779(CHEMBL3758577)
Affinity DataEC50:  0.562nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
University Of California At Los Angeles

Curated by ChEMBL
LigandPNGBDBM50500784(CHEMBL4299242)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at recombinant human NMU1 expressed in HEK293 cells assessed as change in intracellular calcium flux by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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