Affinity DataIC50: 1nMAssay Description:Inhibition of placental sulphatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of human placental microsomal aromatase using testosterone as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of aromatase in human MCF7 cells using [1beta-3H]androstenedione as substrate measured after 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 192nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 202nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 259nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of sulphatase in human MCF7 cells assessed as inhibition of E1-STS activityMore data for this Ligand-Target Pair
Affinity DataIC50: 387nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 539nMAssay Description:Displacement of fluoromone TM from recombinant human ERalpha after 2 hrs by fluorescence polarization analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of aromatase (unknown origin) preincubated for 10 mins in presence of NADPH generating system followed by addition of dibenzylfluorescein ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of aromatase in human MCF7 cells using [1beta-3H]androstenedione as substrate measured after 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of aromatase (unknown origin) preincubated for 10 mins in presence of NADPH generating system followed by addition of dibenzylfluorescein ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of aromatase (unknown origin) preincubated for 10 mins in presence of NADPH generating system followed by addition of dibenzylfluorescein ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab
Curated by ChEMBL
Central University Of Punjab
Curated by ChEMBL
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
Affinity DataIC50: 2.66E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab
Curated by ChEMBL
Central University Of Punjab
Curated by ChEMBL
Affinity DataIC50: 3.09E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
Affinity DataIC50: 3.17E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab
Curated by ChEMBL
Central University Of Punjab
Curated by ChEMBL
Affinity DataIC50: 3.65E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
Affinity DataIC50: 5.12E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.08E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.11E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Central University Of Punjab
Curated by ChEMBL
Central University Of Punjab
Curated by ChEMBL
Affinity DataIC50: 7.35E+4nMAssay Description:Inhibition of His6-tagged Src kinase domain (unknown origin) using AEEEIYGEFEAKKKK as substrate preincubated for 10 mins followed by substrate/ATP ad...More data for this Ligand-Target Pair
Affinity DataIC50: 3.56E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.82E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.87E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair