Affinity DataKi: 0.0300nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0850nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]DPCPX from A1 adenosine receptor (unknown origin) expressed in CHO cell membrane incubated for 60 mins at room temperature by NXT...More data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in Wistar Han rat liver membrane assessed as inhibition constant incubated for 120 minsMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant adenosine A2B receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]OSIP339391 from human recombinant Adenosine A2B receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human recombinant A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human recombinant A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to sigma 2 receptor in human MCF7 cells assessed as displacement of compound by measuring inhibition constant of DTG incubated for 1...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 0.680nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]HZ241385 from human A2AAR expressed in HeLa cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysi...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]HZ241385 from human A2AAR expressed in HeLa cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysi...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes assessed as inhibition constant by Wallac 1450 MicroBeta liqu...More data for this Ligand-Target Pair
Ligand Info
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]SCH-58261 from A2A adenosine receptor (unknown origin) expressed in HEK cell membrane incubated for 60 mins at room temperature b...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPCPX from A1 adenosine receptor (unknown origin) expressed in CHO cell membrane incubated for 60 mins at room temperature by NXT...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cell membrane incubated for 60 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.51nMAssay Description:Binding affinity to recombinant human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.55nMAssay Description:Binding affinity to recombinant human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]HZ241385 from human A2AAR expressed in HeLa cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysi...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cell membrane incubated for 60 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]4-(2-[7-amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol from human adenosine A2A receptor expressed ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM2421385 from adenosine A2A receptor expressed in human HeLa cell membranes incubated for 30 mins by scintillation counting meth...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]HZ241385 from human A2AAR expressed in HeLa cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysi...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385 from human Adenosine A2A receptor expressed in HeLa cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385/[125I]IABOPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385 from human recombinant A2A receptor expressed in human HeLa cell membranes incubated for 30 mins by radioligand binding ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]ZM241385 from human recombinant A2A receptor expressed in human HeLa cell membranes incubated for 30 mins by radioligand binding ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.91nMAssay Description:Binding affinity to recombinant human adenosine A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]IABOPX from human recombinant Adenosine A2B receptor expressed in HEK293 cells after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to recombinant human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in human HeLa cell membranes incubated for 180 mins by radioligand binding competition assa...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]NECA from human A3 receptor expressed in human HeLa cell membranes incubated for 180 mins by radioligand binding competition assa...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human A2B receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De Santiago De Compostela
Curated by ChEMBL
Universidade De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cell membrane incubated for 60 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.14nMAssay Description:Binding affinity to recombinant human adenosine A2B receptorMore data for this Ligand-Target Pair