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Found 400 with Last Name = 'tian' and Initial = 'r'
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094971(CHEMBL3589383)
Affinity DataKi:  12nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094970(CHEMBL3589385)
Affinity DataKi:  14nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094973(CHEMBL3589381)
Affinity DataKi:  18nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50425732(ENZALUTAMIDE | US10053433, FC 4.129 | US10806720, ...)
Affinity DataKi:  28nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094974(CHEMBL3589380)
Affinity DataKi:  34nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094975(956104-40-8 | ARN-509 | JNJ-56021927 | US10053433,...)
Affinity DataKi:  35nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094966(CHEMBL3588961)
Affinity DataKi:  41nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094957(CHEMBL3588965)
Affinity DataKi:  43nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094967(CHEMBL3588960)
Affinity DataKi:  68nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094958(CHEMBL3588959)
Affinity DataKi:  95nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094969(CHEMBL3589387)
Affinity DataKi:  126nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373038(CHEMBL407567)
Affinity DataKi:  150nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301283((R)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMBL5...)
Affinity DataKi:  160nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM18525(Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301281((+/-)-2-benzyl-5,5,5-trifluoro-4-oxopentanoic acid...)
Affinity DataKi:  200nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094972(CHEMBL3589382)
Affinity DataKi:  215nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094963(CHEMBL3588964)
Affinity DataKi:  236nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094960(CHEMBL3589390)
Affinity DataKi:  257nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Henan University

Curated by ChEMBL
LigandPNGBDBM50443692(CHEMBL3093837)
Affinity DataKi:  386nMAssay Description:Mixed-type inhibition of electric eel AChE using acetylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition by Linewea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301282((+/-)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMB...)
Affinity DataKi:  430nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373036(CHEMBL259621)
Affinity DataKi:  450nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094959(CHEMBL3589391)
Affinity DataKi:  482nMAssay Description:Partial agonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094964(CHEMBL3588963)
Affinity DataKi:  515nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094961(CHEMBL3588968)
Affinity DataKi:  576nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094962(CHEMBL3588967)
Affinity DataKi:  585nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373037(CHEMBL261332)
Affinity DataKi:  790nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Alla Chem

Curated by ChEMBL
LigandPNGBDBM50094965(CHEMBL3588962)
Affinity DataKi:  798nMAssay Description:Antagonist activity at androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373039(CHEMBL407566)
Affinity DataKi:  2.08E+3nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301280((+/-)-2-benzyl-5-bromo-4-oxopentanoic acid | CHEMB...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301284((S)-2-benzyl-5-nitro-4-oxopentanoic acid | CHEMBL5...)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373035(CHEMBL259221)
Affinity DataKi:  6.26E+4nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50373037(CHEMBL261332)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of CPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase A1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL
LigandPNGBDBM50301279((+/-)-2-benzyl-4-oxopentanoic acid | CHEMBL568460)
Affinity DataKi:  2.07E+5nMAssay Description:Inhibition of Carboxypeptidase A assessed as amount of Cl-CPL consumed by UV spectrometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547628(CHEMBL4753603)
Affinity DataIC50:  0.00100nMAssay Description:Inhibition of HCV genotype 2a NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by bright Glo-luci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547638(CHEMBL4782728)
Affinity DataIC50:  0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547630(CHEMBL4758660)
Affinity DataIC50:  0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547646(CHEMBL4780371)
Affinity DataIC50:  0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547634(CHEMBL4747100)
Affinity DataIC50:  0.00100nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547637(CHEMBL4745761)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547629(CHEMBL4763617)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547635(CHEMBL4798433)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547636(CHEMBL4744064)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547650(CHEMBL4797491)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547643(CHEMBL4764688)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547627(CHEMBL4755593)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547640(CHEMBL4746579)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547631(CHEMBL4798211)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547639(CHEMBL4744183)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547642(CHEMBL4780002)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 5A(Hepatitis C virus)
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50547649(CHEMBL4793304)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of HCV genotype 1b NS5A infected in Huh7 cells assessed as reduction in viral replication incubated 3 days and measured by Celltiter Glo a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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