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Found 379 with Last Name = 'toogood-johnson' and Initial = 'i'
TargetCaspase-3(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  3nMAssay Description:Inhibition of caspase3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347034(CHEMBL1796096)
Affinity DataIC50:  5nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347036(CHEMBL1796098)
Affinity DataIC50:  6nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347040(CHEMBL1796103)
Affinity DataIC50:  7nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347047(CHEMBL1796230)
Affinity DataIC50:  8nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347046(CHEMBL1796228)
Affinity DataIC50:  9nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347021(CHEMBL1796080)
Affinity DataIC50:  9nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347041(CHEMBL1796105)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347038(CHEMBL1796101)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347044(CHEMBL1796226)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347035(CHEMBL1796097)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420459(CHEMBL2086528)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347050(CHEMBL1796104)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347043(CHEMBL1796225)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  11nMAssay Description:Inhibition of thrombin activated human TG3 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420454(CHEMBL2086544)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420451(CHEMBL2086541)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Mus musculus)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420459(CHEMBL2086528)
Affinity DataIC50:  16nMAssay Description:Inhibition of mouse recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant TG1 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347042(CHEMBL1796106)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347039(CHEMBL1796102)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347048(CHEMBL1796229)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347028(CHEMBL1796089)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420515(CHEMBL2086523)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420471(CHEMBL2086530)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420468(CHEMBL2086524)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420452(CHEMBL2086542)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347037(CHEMBL1796099)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347020(CHEMBL1796079)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347045(CHEMBL1796227)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347033(CHEMBL1796095)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420463(CHEMBL2086480)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420467(CHEMBL2086521)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420518(CHEMBL2086531)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420469(CHEMBL2086525)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420503(CHEMBL2086505)
Affinity DataIC50:  39nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347049(CHEMBL1796083)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420470(CHEMBL2086526)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420519(CHEMBL2086519)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420464(CHEMBL2086506)
Affinity DataIC50:  46nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347026(CHEMBL1796087)
Affinity DataIC50:  50nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420457(CHEMBL2086890)
Affinity DataIC50:  51nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420443(CHEMBL2086532)
Affinity DataIC50:  52nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420504(CHEMBL2086507)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420510(CHEMBL2086515)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420517(CHEMBL2086529)
Affinity DataIC50:  55nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420516(CHEMBL2086527)
Affinity DataIC50:  57nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50347022(CHEMBL1796081)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli nickel containing peptide deformylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420511(CHEMBL2086516)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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