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Found 50 with Last Name = 'umezawa' and Initial = 'y'
LigandPNGBDBM50475041(CHEMBL181131 | TP-104)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475039(CHEMBL181025 | TP-103)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475046(CHEMBL360654 | TP-108)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475038(CHEMBL181235 | TP-102)
Affinity DataIC50:  27nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475036(CHEMBL361462 | TP-110)
Affinity DataIC50:  27nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475040(CHEMBL178839)
Affinity DataIC50:  37nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  68nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
LigandPNGBDBM50475044(CHEMBL362470 | TP-107)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475042(TYROPEPTIN A)
Affinity DataIC50:  140nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475045(CHEMBL180032 | TP-106)
Affinity DataIC50:  190nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50:  330nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475039(CHEMBL181025 | TP-103)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475043(CHEMBL2371767)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475041(CHEMBL181131 | TP-104)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360804(CHEMBL1934668)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327305(CHEMBL1258849 | N,N-dimethyl-1-(4-(((2-phenyl-2H-1...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475040(CHEMBL178839)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475038(CHEMBL181235 | TP-102)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327308(CHEMBL1233973 | LAURYL DIMETHYLAMINE-N-OXIDE | N,N...)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360803(CHEMBL1934667)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
LigandPNGBDBM50475039(CHEMBL181025 | TP-103)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360805(CHEMBL1934669)
Affinity DataIC50:  4.75E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475041(CHEMBL181131 | TP-104)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475042(TYROPEPTIN A)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360806(CHEMBL1934670)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475046(CHEMBL360654 | TP-108)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327308(CHEMBL1233973 | LAURYL DIMETHYLAMINE-N-OXIDE | N,N...)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475043(CHEMBL2371767)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50360802(CHEMBL1710736)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human OSC expressed in Saccharomyces cerevisiae by gas chromatographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327304(1-(4-(((1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol...)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475038(CHEMBL181235 | TP-102)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475040(CHEMBL178839)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475045(CHEMBL180032 | TP-106)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475045(CHEMBL180032 | TP-106)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475035(CHEMBL362804 | TP-109)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327306(CHEMBL1258964 | N-(4-((dimethylamino)methyl)benzyl...)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475044(CHEMBL362470 | TP-107)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475046(CHEMBL360654 | TP-108)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475044(CHEMBL362470 | TP-107)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Homo sapiens (Human))
Institute Of Microbial Chemistry

Curated by ChEMBL
LigandPNGBDBM50327307(4-((dimethylamino)methyl)-N-((1-(4-methoxyphenyl)-...)
Affinity DataIC50:  5.88E+4nMAssay Description:Inhibition of OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475042(TYROPEPTIN A)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50475036(CHEMBL361462 | TP-110)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475036(CHEMBL361462 | TP-110)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50475043(CHEMBL2371767)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed