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Found 82 with Last Name = 'zawadzki' and Initial = 'p'
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508585(CHEMBL4550810)
Affinity DataIC50:  98nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508596(CHEMBL4450084)
Affinity DataIC50:  112nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508606(CHEMBL4452507)
Affinity DataIC50:  122nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508586(CHEMBL4543318)
Affinity DataIC50:  141nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508584(CHEMBL4563315)
Affinity DataIC50:  192nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508602(CHEMBL4451160)
Affinity DataIC50:  222nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508593(CHEMBL4471276)
Affinity DataIC50:  241nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508594(CHEMBL4525991)
Affinity DataIC50:  269nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508610(CHEMBL4561737)
Affinity DataIC50:  313nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508592(CHEMBL4535071)
Affinity DataIC50:  350nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508603(CHEMBL4525206)
Affinity DataIC50:  388nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508595(CHEMBL4584382)
Affinity DataIC50:  494nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508601(CHEMBL4476804)
Affinity DataIC50:  540nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508604(CHEMBL4538177)
Affinity DataIC50:  575nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508612(CHEMBL4454199)
Affinity DataIC50:  599nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508589(CHEMBL4466246)
Affinity DataIC50:  638nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508587(CHEMBL4517341)
Affinity DataIC50:  707nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508600(CHEMBL4579783)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508609(CHEMBL1419805)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508613(CHEMBL4564918)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508614(CHEMBL4577252)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508605(CHEMBL4467842)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508608(CHEMBL4461952)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508599(CHEMBL4445131)
Affinity DataIC50:  4.13E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508611(CHEMBL3975306)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508607(CHEMBL4563640)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM49075(2-(allylamino)-4-amino-5-(2,2-dimethylpropanoyl)-3...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508598(CHEMBL4446294)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508597(CHEMBL4560455)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508591(CHEMBL4460795)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508590(CHEMBL4585980)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508588(CHEMBL4471795)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508583(CHEMBL4466827)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508582(CHEMBL4468259)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508615(CHEMBL4549181)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMaternal embryonic leucine zipper kinase(Homo sapiens (Human))
Selvita

Curated by ChEMBL
LigandPNGBDBM50508581(CHEMBL4544167)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human MELK expressed in Escherichia coli using ZIPtide as substrate measured after 0.5 hrs by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323546(4-((E)-styryl)-pyrimidin-2-ylamine | CHEMBL1209431)
Affinity DataIC50: >1.00E+4nMAssay Description:Negative allosteric modulation of rat mGluR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323546(4-((E)-styryl)-pyrimidin-2-ylamine | CHEMBL1209431)
Affinity DataIC50: >3.00E+4nMAssay Description:Negative allosteric modulation of human mGluR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323546(4-((E)-styryl)-pyrimidin-2-ylamine | CHEMBL1209431)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323546(4-((E)-styryl)-pyrimidin-2-ylamine | CHEMBL1209431)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of rat mGluR4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323548(CHEMBL1209433 | N,N-dimethyl-4-styrylpyrimidin-2-a...)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323549(CHEMBL1209434 | N-(4-styrylpyrimidin-2-yl)methanes...)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323550(2-methyl-4-styrylpyrimidine | CHEMBL1209435)
Affinity DataEC50:  6.90E+3nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323551(2-phenyl-4-styrylpyrimidine | CHEMBL1209436)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323552(4-styrylpyrimidine-2-thiol | CHEMBL1209437)
Affinity DataEC50:  7.80E+3nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323553(4-methyl-6-styrylpyrimidin-2-amine | CHEMBL1209438)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323554(5-methyl-4-styrylpyrimidin-2-amine | CHEMBL1209514)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323555(4,5-dimethyl-6-styrylpyrimidin-2-amine | CHEMBL120...)
Affinity DataEC50:  1.60E+3nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323556(6-styrylpyrimidine-2,4-diamine | CHEMBL1209516)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50323557(2-amino-6-styrylpyrimidin-4-ol | CHEMBL1209517)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human mGluR4 expressed in CHO-K1 cells assessed as decrease in forskolin-induced intracellular cAMP accumulation af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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