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Found 93 with Last Name = 'zechel' and Initial = 'c'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112996(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112986(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113000(3-(2-{[2-(3-Benzyl-ureido)-oxazole-5-carbonyl]-ami...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112985(3-(2-{[2-(3-Benzyl-ureido)-thiazole-4-carbonyl]-am...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113007(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122205((R)-4-{4-[3-(1H-Benzoimidazol-2-ylamino)-propylami...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122205((R)-4-{4-[3-(1H-Benzoimidazol-2-ylamino)-propylami...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112993((S)-2-Benzyloxycarbonylamino-3-(2-{[5-(3-benzyl-ur...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112988(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.5nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113013(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  0.900nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122204((S)-3-{4-[4-(1H-Benzoimidazol-2-ylamino)-piperidin...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122219((R)-4-{4-[4-(1H-Benzoimidazol-2-ylamino)-piperidin...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122198((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122192((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of alphaIIb-beta3 integrin binding to fibrinogen in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122195((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122227((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112987(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113010((S)-2-Benzyloxycarbonylamino-3-(2-{[2-(3-benzyl-ur...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112990(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-amino...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113015(3-(2-{[5-(3-Benzyl-ureido)-thiophene-3-carbonyl]-a...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122225((S)-2-Benzyloxycarbonylamino-3-{5-methyl-2-oxo-4-[...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122222((R)-3-Benzyloxycarbonylamino-4-{4-[3-(1H-imidazol-...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112991((R)-2-Benzyloxycarbonylamino-3-(3-{[5-(3-benzyl-ur...)
Affinity DataIC50:  3.10nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50114263(((R)-2-{(S)-2-[(5-Carbamimidoyl-thiophen-2-ylmethy...)
Affinity DataIC50:  3.60nMAssay Description:In vitro Inhibitory concentration against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122216((R)-3-Benzyloxycarbonylamino-4-{4-[2-(1H-imidazol-...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113011(3-(2-{[2-(3-Benzyl-ureido)-oxazole-5-carbonyl]-ami...)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122228((S)-2-Benzyloxycarbonylamino-3-(4-{[2-(3-benzyl-ur...)
Affinity DataIC50:  4.20nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15471(4-[(1-{[2-oxo-2-(thiophen-3-yl)ethyl]amino}cyclope...)
Affinity DataIC50:  5nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112999((S)-2-Benzyloxycarbonylamino-3-(2-{[5-(3-benzyl-ur...)
Affinity DataIC50:  8.90nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122218((S)-3-{4-[4-(1H-Benzoimidazol-2-yl)-piperidin-1-yl...)
Affinity DataIC50:  9.40nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122220((R)-4-(4-{4-[2-(1H-Benzoimidazol-2-ylamino)-ethyl]...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122198((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122202((S)-2-Benzyloxycarbonylamino-3-{5-methyl-2-oxo-4-[...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122229((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113002(3-(2-{[2-(3-Benzyl-ureido)-oxazole-4-carbonyl]-ami...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122211((S)-3-(4-{4-[2-(1H-Benzoimidazol-2-ylamino)-ethyl]...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113014(3-(2-{[4-(3-Benzyl-ureido)-1-methyl-1H-pyrrole-2-c...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122237((S)-3-(4-{4-[(1H-Benzoimidazol-2-ylamino)-methyl]-...)
Affinity DataIC50:  16nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122214((R)-4-{4-[4-(1H-Benzoimidazol-2-ylamino)-butylamin...)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122203((S)-3-{4-[4-(1H-Benzoimidazol-2-ylmethyl)-piperidi...)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122217((R)-4-{4-[2-(1H-Benzoimidazol-2-ylcarbamoyl)-ethyl...)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122230((R)-3-Benzyloxycarbonylamino-4-{5-methyl-2-oxo-4-[...)
Affinity DataIC50:  36nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Eli Lilly

LigandPNGBDBM15465(4-[(3R)-3-{[2-(3,4-difluorophenyl)-2-oxoethyl]amin...)
Affinity DataIC50:  39nMpH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122231((R)-3-Benzyloxycarbonylamino-4-{4-[4-(3-benzyl-ure...)
Affinity DataIC50:  39nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50112997((R)-3-Benzyloxycarbonylamino-4-(2-{[5-(3-benzyl-ur...)
Affinity DataIC50:  44nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122199((S)-3-{4-[4-(1H-Benzoimidazol-2-ylamino)-butylamin...)
Affinity DataIC50:  47nMAssay Description:Inhibition of alphaIIb-beta3 integrin binding to fibrinogen in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122212((R)-3-Benzyloxycarbonylamino-4-(4-{[2-(3-benzyl-ur...)
Affinity DataIC50:  48nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113006(3-(2-{[5-(3-Benzyl-ureido)-furan-2-carbonyl]-methy...)
Affinity DataIC50:  51nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50122221((S)-3-{4-[3-(1H-Benzoimidazol-2-ylamino)-propylami...)
Affinity DataIC50:  61nMAssay Description:Inhibitory concentration against alphaV-beta3 integrin using vitronectin ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Basf

Curated by ChEMBL
LigandPNGBDBM50113003(3-(2-{[5-(3-Benzyl-ureido)-1H-[1,2,4]triazole-3-ca...)
Affinity DataIC50:  72nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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