TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contraction in presence of TRPV1 an...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 3.98E+3nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 6.31E+3nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.51nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 6.31nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.51nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.51nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 6.31nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as inhibition of capsaicin-induced intracellular calciu...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 0.501nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contraction in presence of TRPV1 an...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 63nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contraction in presence of TRPV1 an...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Lund University
Curated by ChEMBL
Lund University
Curated by ChEMBL
Affinity DataEC50: 398nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contraction in presence of TRPV1 an...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Universidad De Antioquia
Curated by ChEMBL
Universidad De Antioquia
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at human TRPV1 expressed in tetracycline-stimulated HEK293 cells assessed as increase in intracellular calcium levels by fluorimetri...More data for this Ligand-Target Pair