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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
11
hits in this display
Target
Monocarboxylate transporter 1
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
MCT1 activity may be measured using BT-20 breast cancer cells that express high native levels of MCT1, but do not express MCT4 and are known to those...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Malignant T-cell-amplified sequence 1
(Homo sapiens (human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
MCT1 activity may be measured using BT-20 breast cancer cells that express high native levels of MCT1, but do not express MCT4 and are known to those...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 440nM
Assay Description:
MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 440nM
Assay Description:
MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 440nM
Assay Description:
MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 860nM
Assay Description:
NCI-H358 lung adenocarcinoma cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 860nM
Assay Description:
NCI-H358 lung adenocarcinoma cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 860nM
Assay Description:
NCI-H358 lung adenocarcinoma cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 4
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 860nM
Assay Description:
NCI-H358 lung adenocarcinoma cells may be used to measure MCT4 activity in cells with high native levels of MCT4 and low levels of MCT1 and are known...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 1
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.20E+3nM
Assay Description:
MCT1 activity may be measured using BT-20 breast cancer cells that express high native levels of MCT1, but do not express MCT4 and are known to those...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Monocarboxylate transporter 1
(Homo sapiens (Human))
Vettore
US Patent
Ligand
BDBM345271
(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.20E+3nM
Assay Description:
MCT1 activity may be measured using BT-20 breast cancer cells that express high native levels of MCT1, but do not express MCT4 and are known to those...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI