TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 7.0 T: 2°CAssay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in DMG buffer (50 mM DMG, pH 7.0, 1 mM EDTA, 150 mM NaCl, 2 mM DTT, 0.1 ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of DUSP22 (unknown origin) pre-incubated for 20 mins followed by fluorescence substrate addition and measured after 120 mins by DiFMUP ass...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 5.55E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 8.05E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 8.36E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 8.39E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >1.00E+4nMpH: 7.0Assay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in 3,3-dimethylglutarate buffer (50 mM 3,3-dimethylglutarate, pH 7.0, 1 ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant VHX (unknown origin) using OMFP as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >5.00E+4nMpH: 6.0 T: 2°CAssay Description:PTP assay were conducted at 25 C in 96-well plates. Reaction rates were determined using a Variokan plate reader from Thermo Electron. For assay pH...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research and Technology
US Patent
Indiana University Research and Technology
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair