TargetHistone acetyltransferase p300(Homo sapiens (Human))
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant His-tagged HAT p300 expressed in Sf21-Baculovirus systemMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant His-tagged p300 HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of TIP60 in human HeLa cell extracts by ELISAMore data for this Ligand-Target Pair
TargetGlyceraldehyde-3-phosphate dehydrogenase, glycosomal(Trypanosoma cruzi)
Universidade Federal De S£O Carlos
Curated by ChEMBL
Universidade Federal De S£O Carlos
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant glycosomal GAPDH expressed in Escherichia coli using GAPDH and D-glyceraldehyde-3-phosphateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of PCAF (unknown origin) using histone H3/[acetyl-3H]-acetyl coenzyme A as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human MOF expressed in Escherichia coli BL21(DE3) cells using [14C]AC-CoA and histone H4 as substrate after 5 mins by scintillation cou...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of human recombinant His-tagged Tip60 expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate after 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of soybean lipoxygenase-1More data for this Ligand-Target Pair
TargetDecaprenyl diphosphate synthase(Mycobacterium tuberculosis H37Rv)
University of California San Diego
University of California San Diego
Affinity DataIC50: 2.80E+5nMpH: 7.5Assay Description:We screened an in-house library of 53 compounds using trans-FPP as substrate. Briefly, the condensation of IPP and GPP, FPP, or cis-FPP catalyzed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.75E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.67E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human recombinant histone deacetylase PCAF by ELISAMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
The Institute Of Cancer Research
Curated by ChEMBL
The Institute Of Cancer Research
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+6nMAssay Description:Concentration required for its inhibitory activity against Escherichia coli JT4(TEM1) class A beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.21E+6nMAssay Description:Concentration required for its inhibitory activity against Escherichia coli K12(PSE4) class A beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.08E+6nMAssay Description:Concentration required for its inhibitory activity against Enterobacter cloacae P99 class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+7nMAssay Description:Concentration required for its inhibitory activity against Pseudomonas aeruginosa class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.29E+7nMAssay Description:Concentration required for its inhibitory activity against Escherichia coli K12(OXA1) class D beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.05E+7nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair