Affinity DataIC50: 9nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced inhibition of calcium fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as inhibition of MCP1-induced inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 249nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 254nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 284nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 301nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 328nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 438nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 744nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 928nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.64E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.97E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.42E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.48E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.41E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.78E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.15E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.61E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.74E+3nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [125I]MCP-1 from CCR2 in human PBMC by radioligand displacement assayMore data for this Ligand-Target Pair