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Found 7 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-2' and Ligand = 'BDBM50008859'
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of sirtuin 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of Phosphodiesterase 2 from pig coronary arteryMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of SIRT-2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of recombinant human full length SIRT2 using fluorescent ZMAL as substrate after 4 hrs by homogeneous fluorescent deacetylase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human recombinant SIRT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50008859(CHEMBL3222141)
Affinity DataIC50:  1.55E+7nMAssay Description:Inhibition of SIRT2 (unknown origin) using fluorogenic deacetylase substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed