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Found
1
Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase tankyrase-1' and Ligand = 'BDBM318028'
Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
Eli Lilly
US Patent
Ligand
BDBM318028
(2-[4-[(2- Methoxyphenyl)methyl]piperazin- 1-yl]-8-...)
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Affinity Data
IC50: 18.4nM
Assay Description:
The enzymatic activity of hTNKS1 and hTNKS2 is assessed using an enzyme-linked immunosorbent assay (ELISA) which detects poly ADP ribose incorporated...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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