Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for monomerid = 31587
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50:  2.30nMpH: 7.5 T: 2°CAssay Description:Human GSK-3beta was expressed as the N-terminal FLAG-tagged protein using a baculovirus expression system. The kinase assay was was conducted in a 96...More data for this Ligand-Target Pair
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TargetProtein kinase C theta type(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50:  3.50E+3nMAssay Description:Assays for serine/threonine kinases using radiolabeled [gamma-33P] ATP (GE Healthcare, Piscataway, NJ) were performed in 96 well plates. Prior to the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50:  4.60E+3nMAssay Description:Assays for serine/threonine kinases using radiolabeled [gamma-33P] ATP (GE Healthcare, Piscataway, NJ) were performed in 96 well plates. Prior to the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50:  8.10E+3nMAssay Description:Assays for serine/threonine kinases using radiolabeled [gamma-33P] ATP (GE Healthcare, Piscataway, NJ) were performed in 96 well plates. Prior to the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50: >1.00E+4nMAssay Description:Assays for serine/threonine kinases using radiolabeled [gamma-33P] ATP (GE Healthcare, Piscataway, NJ) were performed in 96 well plates. Prior to the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50: >1.00E+4nMT: 2°CAssay Description:Human p35/ cyclin dependent kinase 5 (CDK5) was purchased from Millipore Corp. (Bedford, MA), which was expressed as N-terminal GST fusion protein us...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed