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Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 1' and Ligand = 'BDBM31587'
TargetMitogen-activated protein kinase kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

LigandPNGBDBM31587(oxadiazole derivative, 20x)
Affinity DataIC50:  8.10E+3nMAssay Description:Assays for serine/threonine kinases using radiolabeled [gamma-33P] ATP (GE Healthcare, Piscataway, NJ) were performed in 96 well plates. Prior to the...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed