Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ki for monomerid = 50337327
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi:  402nMAssay Description:Inhibition of Rock2 after 1 hr using biotinylated longS peptide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi:  3.69E+3nMAssay Description:Inhibition of Pim1 after 1 hr using biotinylated AL1peptide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi: >3.75E+3nMAssay Description:Inhibition of Pak4 after 1 hr using biotinylated L15 peptide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi:  4.27E+3nMAssay Description:Inhibition of GSK3-beta after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi: >4.90E+3nMAssay Description:Inhibition of Aurora kinase 2 after 1 hr using biotinylated kemptide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337327(5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamid...)
Affinity DataKi: >8.88E+3nMAssay Description:Inhibition of KDR after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed