BDBM50337327 5-(1H-indazol-5-yl)-N-methylisoxazole-3-carboxamide::CHEMBL1681795
SMILES CNC(=O)c1cc(on1)-c1ccc2[nH]ncc2c1
InChI Key InChIKey=PYWUGDQVHDHKLX-UHFFFAOYSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50337327
Affinity DataKi: 402nMAssay Description:Inhibition of Rock2 after 1 hr using biotinylated longS peptide as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: 3.69E+3nMAssay Description:Inhibition of Pim1 after 1 hr using biotinylated AL1peptide as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: >3.75E+3nMAssay Description:Inhibition of Pak4 after 1 hr using biotinylated L15 peptide as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 4.27E+3nMAssay Description:Inhibition of GSK3-beta after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: >4.90E+3nMAssay Description:Inhibition of Aurora kinase 2 after 1 hr using biotinylated kemptide as substrateMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataKi: >8.88E+3nMAssay Description:Inhibition of KDR after 1 hrMore data for this Ligand-Target Pair