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Found 2 Enz. Inhib. hit(s) with Target = '[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial' and Ligand = 'BDBM50232913'
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
National Institute Of Biological Science

Curated by ChEMBL
LigandPNGBDBM50232913(CHEMBL4103350)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of recombinant human PDK1 in presence of E1 protein and PDC core E2/E3BP incubated for 10 mins by titration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
National Institute Of Biological Science

Curated by ChEMBL
LigandPNGBDBM50232913(CHEMBL4103350)
Affinity DataIC50:  2.54E+3nMAssay Description:Inhibition of recombinant human PDK1 in presence of E1 protein incubated for 10 mins by titration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed