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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM319627'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Xinjiang Technical Institute of Physics and Chemistry

Curated by ChEMBL
LigandPNGBDBM319627(3-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)ethy...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at 5-HT2A receptor (unknown origin) after 10 mins by calcium 5 dye based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Xinjiang Technical Institute of Physics and Chemistry

Curated by ChEMBL
LigandPNGBDBM319627(3-(2-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)ethy...)
Affinity DataIC50:  25.4nMAssay Description:The 5-HT2A receptor antagonism activity test (The antagonism activity of test compounds on 5-HT2A receptor expressing human recombinant 5-HT2A recept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent