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Found 1 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50161637'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161637((R)-8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-...)
Affinity DataEC50:  220nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2C receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed