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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM29528'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29528(ML10302 scaffold, 9{a;y})
Affinity DataKi:  111nM ΔG°:  -39.7kJ/mole EC50:  4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding studies were performed in buffer contains test compound, [3H]-GR113808, and receptor C6 glial cell membrane preparation. Nonspeci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs

LigandPNGBDBM29528(ML10302 scaffold, 9{a;y})
Affinity DataAssay Description:EC/IC50 was the effective concentration of agonist inhibiting the formation of A-beta fibrils to 50% of the control value. Three independent measurem...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed