Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50240618'
Affinity DataKi: 3.98nMAssay Description:Displacement of [3H]GR113808 from human recombinant 5HT4C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Displacement of [3H]GR113808 from human recombinant 5HT4c receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [N-methyl-3H]GR113808 from human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.31nMAssay Description:Agonist activity at 5HT4 receptor in guinea pig colonic longitudinal muscle/myentric plexus assessed as contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Induction of 5-HT4 receptor-mediated contraction in guinea pig longitudinal muscle myenteric plexusMore data for this Ligand-Target Pair
Affinity DataEC50: 6.31nMAssay Description:Agonist activity at 5HT4 receptor in guinea pig colon assessed as longitudinal muscle plexus contractionMore data for this Ligand-Target Pair