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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 7' and Ligand = 'BDBM21371'
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21371(6-[4-(2-hydroxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21371(6-[4-(2-hydroxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  11.4nM ΔG°:  -47.2kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21371(6-[4-(2-hydroxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  11.4nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed