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Found 2 Enz. Inhib. hit(s) with Target = '72 kDa type IV collagenase' and Ligand = 'BDBM50124122'
Target72 kDa type IV collagenase(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50124122(CHEMBL3622800)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of APMA-activated human recombinant MMP2 incubated for 5 mins using 4-nitrophenylacetate substrate by esterase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50124122(CHEMBL3622800)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition of recombinant human MMP-2 preincubated for 10 mins followed by Mca-PLGL-Dpa-AR-NH2 substrate addition and measured for 5 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed