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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'ADAMTS5' and Ligand = 'BDBM471828'
Target
ADAMTS5
(Rattus norvegicus (Rat))
Galapagos
US Patent
Ligand
BDBM471828
((5S)-5-[(2S)-3-[4- (3,4-difluoro-5- methoxy- pheny...)
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Affinity Data
IC50: 12.5nM
Assay Description:
TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...
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Target Info
PDB
UniProtKB/TrEMBL
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Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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