Affinity DataKi: 6.10nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatum using [3H]NECA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Inhibition of [3H]NECA binding to adenosine A2 receptor from rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatal membranes using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataEC50: 681nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair