Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50067079'
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067079(1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-ethan...)
Affinity DataKi:  660nMAssay Description:Binding affinity of the compound was determined by its ability to displace [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067079(1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-ethan...)
Affinity DataKi:  6.60E+5nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067079(1-Phenyl-2-(3-pyridin-2-yl-isoquinolin-1-yl)-ethan...)
Affinity DataKi:  6.60E+5nMAssay Description:Tested for antagonist activity by displacement of specific [125I]-AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed