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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50344057'
TargetAdenosine receptor A3(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50344057(8-Ethoxy-3-(4'-methoxyphenyl)coumarin | CHEMBL1777...)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cells measured by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50344057(8-Ethoxy-3-(4'-methoxyphenyl)coumarin | CHEMBL1777...)
Affinity DataKi:  5.32E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50344057(8-Ethoxy-3-(4'-methoxyphenyl)coumarin | CHEMBL1777...)
Affinity DataIC50:  2.95E+4nMAssay Description:Antagonist activity at human adenosine receptor A3 expressed in CHO cells assessed as suppression of NECA-induced decrease of cAMP accumulation by Gl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed