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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM86761'
TargetAdenosine receptor A3(Homo sapiens (Human))
Hokkaido University

Curated by PDSP Ki Database
LigandPNGBDBM86761(CAS_35920-39-9 | NECA | NSC_448222)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Hokkaido University

Curated by PDSP Ki Database
LigandPNGBDBM86761(CAS_35920-39-9 | NECA | NSC_448222)
Affinity DataKi:  73nM ΔG°:  -40.7kJ/molepH: 7.4 T: 2°CAssay Description:Aliquots of cell membranes (90 ug) were incubated at 25 °C for 180 min in 500 uL of binding buffer (50 mM Tris-HCl, 5 mM MgCl2, 1 mM EDTA, 2 un...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed