Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor' and Ligand = 'BDBM50001888'
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Solvay Pharma
Curated by ChEMBL
Solvay Pharma
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Solvay Pharma
Curated by ChEMBL
Solvay Pharma
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:The compound was tested for its binding affinity towards alpha-1 adrenergic receptor by displacing [3H]WB-4101 radioligand in rat cerebral cortexcMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Solvay Pharma
Curated by ChEMBL
Solvay Pharma
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Solvay Pharma
Curated by ChEMBL
Solvay Pharma
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Ability to bind at Alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair