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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A/Alpha-2A adrenergic receptor' and Ligand = 'BDBM50027226'
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site A using [3H]clonidineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50:  3nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site B using [3H]-clonidineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50:  100nMAssay Description:In vitro binding affinity of alpha-adrenoceptor by interacting with high affinity, [3H]serotonin from calf caudate nucleusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed