Affinity DataKi: 19nMAssay Description:Binding assay using 5-HT2A, Dopamine D2, SERT, αA1, 5-HT2C and H1 Receptors.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Centro De InvestigacióN Grupo Ferrer
Curated by ChEMBL
Centro De InvestigacióN Grupo Ferrer
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity measured at the Alpha-1A adrenergic receptor by the inhibition of [3H]-prazosin binding to rat cortex using unlabeled WB-4101 for no...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(CALF)
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Institut De Chimie Pharmaceutique Albert Lespagnol
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Affinity towards Alpha-1A adrenergic receptor in membranes from bovine frontal cortex using [3H]-prazosinMore data for this Ligand-Target Pair