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Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM9463'
TargetAromatase(Homo sapiens (Human))
Universidade De Coimbra

Curated by ChEMBL
LigandPNGBDBM9463(3-(1H-Imidazol-1-ylmethyl)-5H-indeno[1,2-c]pyridaz...)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universidade De Coimbra

Curated by ChEMBL
LigandPNGBDBM9463(3-(1H-Imidazol-1-ylmethyl)-5H-indeno[1,2-c]pyridaz...)
Affinity DataIC50:  2.66E+4nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta, 2beta-3H] testosterone or [1beta-3H] androstenedione during aroma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed