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Found 3 Enz. Inhib. hit(s) with Target = 'Aryl hydrocarbon receptor' and Ligand = 'BDBM23936'
TargetAryl hydrocarbon receptor(Oryctolagus cuniculus (rabbit))
Institut Claudius Regaud

LigandPNGBDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  0.200nM ΔG°:  -51.5kJ/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to AhR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  2.00E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article