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Found 3 Enz. Inhib. hit(s) with Target = 'Aurora kinase A' and Ligand = 'BDBM92846'
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92846(Bisanilinopyrimidine, 12d | US9249124, 62)
Affinity DataIC50:  3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92846(Bisanilinopyrimidine, 12d | US9249124, 62)
Affinity DataIC50:  3nMpH: 7.4 T: 2°CAssay Description:Reactions were carried out at room temperature in 15 mM HEPES buffer (pH 7.4) containing 20 mM NaCl, 1 mM EGTA, 0.02% Tween 20, 10 mM MgCl2, 5% (v/v)...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92846(Bisanilinopyrimidine, 12d | US9249124, 62)
Affinity DataIC50: >1.00E+4nMT: 2°CAssay Description:Specifically, MDA-MB-468 cells (American Type Culture Collection) were maintained in Dulbecco's modified Eagle's medium (DMEM) plus 10% fetus bovine ...More data for this Ligand-Target Pair
In DepthDetails US Patent