Found 2 Enz. Inhib. hit(s) with Target = 'Aurora kinase B/Inner centromere protein' and Ligand = 'BDBM209861'
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
Nirma University
Curated by ChEMBL
Nirma University
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Inhibition of Aurora B/INCENP (unknown origin) assessed as affinity constant pre-incubated for 1 hr followed by FL-PKAtide substrate and ATP additionMore data for this Ligand-Target Pair
TargetAurora kinase B/Inner centromere protein(Homo sapiens (Human))
Nirma University
Curated by ChEMBL
Nirma University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of Aurora B/INCENP (unknown origin) pre-incubated for 1 hr followed by FL-PKAtide substrate and ATP additionMore data for this Ligand-Target Pair