Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50209745'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50209745((R)-N-((R)-7-((tert-butylamino)methyl)chroman-4-yl...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50209745((R)-N-((R)-7-((tert-butylamino)methyl)chroman-4-yl...)
Affinity DataIC50:  9.90nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHOD cellsassessed as effect on DAK-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed