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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-lactamase OXA-1' and Ligand = 'BDBM50021954'
TargetBeta-lactamase OXA-1(Escherichia coli (Enterobacteria))TBA
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibitory activity against Escherichia coli HA209 Class-V OXA-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase OXA-1(Escherichia coli (Enterobacteria))TBA
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory activity against Beta-lactamase type OXA1 (penicillinase) from E. coli OXA1 using ampicillin (40 uM) as a substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed