Found 11 Enz. Inhib. hit(s) with Target = 'Broad substrate specificity ATP-binding cassette transporter ABCG2' and Ligand = 'BDBM50379211'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in HEK293 cells by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux after 30 mins by FACS methodMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human ABCG2 expressed in Sf9 insect cell membranes assessed as inhibition of quercetin-stimulated ATPase activity after 30 mins by colo...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataIC50: 707nMAssay Description:Inhibition of ABCG2 in topotecan-cultured human MCF7 cells using Hoechst 33342 as substrate measured after 2 hrs by fluorescence assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Inhibition of ABCG2-mediated mitoxantrone efflux in mitoxantrone-selected human H460 cells after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 1.30E+8nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as increase in mitoxantrone accumulation incubated for 30 mins by flow cytome...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Inhibition of ABCG2 (unknown origin) in HEK293 cells assessed as maximal inhibition of mitoxantrone efflux by fluorescence based flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 94nMAssay Description:Inhibition of ABCG2 (unknown origin) transfected in HEK293 cells assessed as inhibition of mitoxantrone efflux after 30 mins by flow cytometry relati...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Inhibition of ABCG2 (unknown origin) transfected in HEK293 cells assessed as inhibition of mitoxantrone efflux at 5 uM after 30 mins in presence of 0...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Cnrs/Universit£
Curated by ChEMBL
Cnrs/Universit£
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Inhibition of ABCG2 (unknown origin)-mediated mitoxantrone efflux expressed in HEK293 cells after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair