Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50559308'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg
Curated by ChEMBL
Albert-Ludwigs-Universit£T Freiburg
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg
Curated by ChEMBL
Albert-Ludwigs-Universit£T Freiburg
Curated by ChEMBL
Affinity DataKd: 260nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair