Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [352-457]' and Ligand = 'BDBM220664' 
Affinity DataKi: 1.20nM ΔG°: -50.9kJ/molepH: 6.0 T: 2°CAssay Description:A time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used to determine the affinities of compounds of the Examples listed in Ta...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 15.5nMAssay Description:Compound dilution series were prepared in DMSO via an approximately 3-fold serial dilution. Compound dilutions were added directly into white, low-vo...More data for this Ligand-Target Pair
