Found 7 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 5' and Ligand = 'BDBM50339033'
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at CCR5 assessed as inhibition of receptor internalizationMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at CCR5 in IL-10 stimulated human PBMC cells assessed as MIP-1beta induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at CCR5 assessed as inhibition of ERK phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity to CCR5More data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 in IL-10-stimulated human monocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at CCR5 assessed as inhibition of intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Activation of CCR5 in human PBMC cellsMore data for this Ligand-Target Pair