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Found 2 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 3' and Ligand = 'BDBM50200679'
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50200679(CHEMBL3916901)
Affinity DataIC50:  74nMAssay Description:Antagonist activity at human Galphai4qi4-coupled CXCR3A expressed in engineered CHO cells assessed as inhibition of IP-10-induced calcium mobilizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50200679(CHEMBL3916901)
Affinity DataIC50:  403nMAssay Description:Displacement of [125I]-CXCL10 from human recombinant CXCR3 transfected in Flp-In-CHO cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed