Affinity DataKi: 7nMAssay Description:The binding affinity against calpain.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity evaluated against recombinant human calpain 1More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against Calpain 1 in platelets.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of calpain (unknown origin) using Suc-LY-AMC as fluorogenic substrate after 60 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 297nMAssay Description:Inhibition of human erythrocytes mu-calpain using Pep1 as substrate incubated for 30 mins under shaking condition in presence of CaCl2 by fluorescenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against calpain.Checked by AuthorMore data for this Ligand-Target Pair