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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM239073'
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239073(US9416103, CP-55,940)
Affinity DataKi:  0.370nM ΔG°:  -53.8kJ/moleT: 2°CAssay Description:Competition receptor binding was performed as previously described [Shoemaker et al., J. Pharmacol. Exp. Ther., 314:868-75]. Briefly, 50 μg of mou...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
University of Arkansas

US Patent
LigandPNGBDBM239073(US9416103, CP-55,940)
Affinity DataEC50:  7.5nMT: 2°CAssay Description:[35S]GTPγS binding was performed as previously described [Brents et al., PLoS One, 6:e21917]. Briefly, 25 μg of mouse brain homogenates were...More data for this Ligand-Target Pair
In DepthDetails US Patent