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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50292278'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataIC50:  120nMAssay Description:Neutral antagonist activity at human CB2 assessed as restoration of forskolin-induced cAMP formation preincubated for 15 mins followed by forskolin a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataIC50:  120nMAssay Description:Inhibition of very late antigen-4 alpha4-beta1 (VLA-4), I-VCAM-Ig as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed