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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50463775'
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50463775(CHEMBL4240671)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CP-55,940 from recombinant mouse Cb2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50463775(CHEMBL4240671)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55,940 from recombinant human Cb2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50463775(CHEMBL4240671)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant human Cb2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP levelsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed