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Found 1 Enz. Inhib. hit(s) with Target = 'Chloroquine resistance transporter' and Ligand = 'BDBM50017696'
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50017696((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed